SCHEMBL12193576

SCHEMBL12193576

Nc1ccc2[nH]nc(-c3ccc(F)c(F)c3)c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 4/20 0.54
AXL P30530 2/20 0.52
MAPK1 P28482 3/20 0.49
MAP2K4 P45985 3/20 0.49
MAPKAPK2 P49137 3/20 0.49
MAPKAPK3 Q16644 3/20 0.49
MAPK6 Q16659 3/20 0.49
AURKA O14965 1/20 0.49
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48
GSK3B P49841 1/20 0.43
JAK2 O60674 2/20 0.43
NOTUM Q6P988 1/20 0.42
IDO1 P14902 1/20 0.42
FGFR1 P11362 1/20 0.42
FGFR2 P21802 1/20 0.42
WNT1 P04628 1/20 0.42
DYRK1A Q13627 1/20 0.42
NTRK1 P04629 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2473158 0.84 AXL (0.52) AXLMAPK1MAP2K4MAPKAPK2MAPKAPK3
SCHEMBL4225769 0.84 MAP2K4 (0.47) TRPA1AXLMAPK1MAP2K4MAPKAPK2
SCHEMBL2469031 0.84 AXL (0.55) AXLMAPK1MAP2K4MAPKAPK2MAPKAPK3
SCHEMBL1663211 0.83 AXL (0.60) AXLMAPK1MAP2K4MAPKAPK2MAPKAPK3
SCHEMBL13854966 0.83 MAP2K4 (0.73) TRPA1AXLMAPK1MAP2K4MAPKAPK2
Hydrochloric Acid SCHEMBL27750634 0.83 AXL (0.54) AXLMAPK1MAP2K4MAPKAPK2MAPKAPK3
SCHEMBL4006856 0.81 AXL (0.55) AXLMAPK1MAP2K4MAPKAPK2MAPKAPK3
SCHEMBL14516332 0.80 AURKA (0.59) AXLMAP2K4AURKAHTR2AHTR2C
SCHEMBL1663041 0.79 AXL (0.50) AXLMAPK1MAP2K4MAPKAPK2MAPKAPK3
SCHEMBL3137122 0.79 MAP2K4 (0.48) TRPA1AXLMAPK1MAP2K4MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966151-B1 POLYCYCLIC INDAZOLE DERIVATIVES THAT ARE ERK INHIBITORS SCHERING CORP (US) 2011-10-05 EP disclosed