SCHEMBL12196129

SCHEMBL12196129

Cc1c[nH]c(C2=NCC(CC(=O)N3CCOCC3)S2)cc(C)cc(Oc2ccc(S(C)(=O)=O)nc2)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 5/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GAA P10253 1/20 0.33
PIK3CD O00329 2/20 0.32
PIK3CA P42336 2/20 0.32
GPR119 Q8TDV5 1/20 0.32
KDM4E B2RXH2 1/20 0.31
GCK P35557 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
POLB P06746 1/20 0.31
ALOX5 P09917 1/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL564342 0.85 FKBP1A (0.35) FKBP1ASMN1; SMN2PIK3CDPIK3CAGCK
SCHEMBL565181 0.84 GCK (0.39) ALDH1A1HPGDKDM4EGCK
SCHEMBL564544 0.80 GCK (0.36) ALDH1A1HPGDPIK3CDPIK3CAGPR119
SCHEMBL564398 0.75 GCK (0.32) GCK
SCHEMBL564085 0.75 GCK (0.34) PIK3CDPIK3CAGPR119GCK
SCHEMBL564086 0.75 GCK (0.34) PIK3CDPIK3CAGPR119GCK
SCHEMBL564470 0.73 GCK (0.32) GCK
SCHEMBL564378 0.71 GCK (0.38) GCK
SCHEMBL565089 0.70 GCK (0.34) GCK
SCHEMBL563538 0.70 GCK (0.39) PIK3CDPIK3CAGPR119GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2371826-A1 NOVEL FUSED RING COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2011-10-05 EP disclosed