SCHEMBL1224740

SCHEMBL1224740

C/C(=C1\C(=O)Nc2ccc(CN3C(=O)COC3=O)cc21)c1cc(CN2CCOCC2)c[nH]1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.49
FGFR1 P11362 1/20 0.49
FGFR2 P21802 1/20 0.49
FGFR3 P22607 1/20 0.49
AXL P30530 1/20 0.49
AKT2 P31751 10/20 0.42
PDPK1 O15530 5/20 0.41
PDK1 Q15118 1/20 0.38
PDGFRB P09619 2/20 0.34
KDR P35968 2/20 0.34
DRD2 P14416 2/20 0.33
DRD4 P21917 2/20 0.33
DRD3 P35462 2/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
MAP4K1 Q92918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1224741 1.00 MET (0.49) METFGFR1FGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260015 0.99 MET (0.48) METFGFR1FGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260014 0.99 MET (0.48) METFGFR1FGFR2FGFR3AXL
SCHEMBL1225733 0.86 MET (0.44) METFGFR1FGFR2FGFR3AXL
SCHEMBL1225734 0.86 MET (0.44) METFGFR1FGFR2FGFR3AXL
SCHEMBL260754 0.86 MET (0.67) METFGFR1FGFR2FGFR3AXL
SCHEMBL260755 0.86 MET (0.67) METFGFR1FGFR2FGFR3AXL
SCHEMBL260141 0.86 AKT2 (0.47) METFGFR1FGFR2FGFR3AXL
SCHEMBL260140 0.86 AKT2 (0.47) METFGFR1FGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260654 0.86 MET (0.44) METFGFR1FGFR2FGFR3AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2281822-B1 New dihydroindolone derivatives, method of preparing same and pharmaceutical compositions containing them SERVIER LAB (FR) 2013-01-16 EP disclosed
EP-2281822-A1 New dihydroindolone derivatives, method of preparing same and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2011-02-09 EP disclosed