SCHEMBL1225440

SCHEMBL1225440

O=C1Nc2ccc(CN3CCOC3=O)cc2C1=Cc1cc(CN2CCCC2)c[nH]1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 3/20 0.61
MET P08581 1/20 0.61
FGFR2 P21802 1/20 0.61
FGFR3 P22607 1/20 0.61
AXL P30530 1/20 0.61
PDPK1 O15530 4/20 0.42
AKT2 P31751 3/20 0.42
NTRK1 P04629 2/20 0.39
FLT3 P36888 3/20 0.38
KDR P35968 5/20 0.37
PDGFRB P09619 2/20 0.37
CSF1R P07333 1/20 0.37
PDGFRA P16234 1/20 0.37
FLT1 P17948 1/20 0.37
LCK P06239 2/20 0.36
FYN P06241 2/20 0.36
YES1 P07947 2/20 0.36
SRC P12931 2/20 0.36
CDK2 P24941 1/20 0.36
MAP4K1 Q92918 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1225437 1.00 FGFR1 (0.61) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260365 0.99 FGFR1 (0.60) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260366 0.99 FGFR1 (0.60) FGFR1METFGFR2FGFR3AXL
SCHEMBL1162294 0.99 FGFR1 (0.60) FGFR1METFGFR2FGFR3AXL
SCHEMBL1162297 0.99 FGFR1 (0.60) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260791 0.98 FGFR1 (0.59) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260792 0.98 FGFR1 (0.59) FGFR1METFGFR2FGFR3AXL
SCHEMBL260188 0.94 FGFR1 (0.69) FGFR1METFGFR2FGFR3AXL
SCHEMBL260189 0.94 FGFR1 (0.69) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260953 0.93 FGFR1 (0.68) FGFR1METFGFR2FGFR3AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2281822-B1 New dihydroindolone derivatives, method of preparing same and pharmaceutical compositions containing them SERVIER LAB (FR) 2013-01-16 EP disclosed
EP-2281822-A1 New dihydroindolone derivatives, method of preparing same and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2011-02-09 EP disclosed