SCHEMBL1225486

SCHEMBL1225486

O=C1Nc2ccc(CN3CCOC3=O)cc2/C1=C/c1c[nH]c(CN2CCOCC2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 3/20 0.51
MET P08581 1/20 0.51
FGFR2 P21802 1/20 0.51
FGFR3 P22607 1/20 0.51
AXL P30530 1/20 0.51
LRRK2 Q5S007 2/20 0.43
FLT3 P36888 1/20 0.43
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
PAK1 Q13153 8/20 0.42
KDR P35968 3/20 0.41
LCK P06239 2/20 0.41
FYN P06241 2/20 0.41
YES1 P07947 2/20 0.41
SRC P12931 2/20 0.41
PDGFRB P09619 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1225487 1.00 FGFR1 (0.51) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260633 0.99 FGFR1 (0.50) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL260632 0.99 FGFR1 (0.50) FGFR1METFGFR2FGFR3AXL
SCHEMBL1225466 0.89 MET (0.40) FGFR1METFGFR2FGFR3AXL
SCHEMBL1225468 0.89 MET (0.40) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL259881 0.88 MET (0.40) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL259880 0.88 MET (0.40) FGFR1METFGFR2FGFR3AXL
Hydrochloric Acid SCHEMBL259879 0.88 MET (0.40) FGFR1METFGFR2FGFR3AXL
SCHEMBL261581 0.86 FGFR1 (0.52) FGFR1METFGFR2FGFR3AXL
SCHEMBL261580 0.86 FGFR1 (0.52) FGFR1METFGFR2FGFR3AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2281822-B1 New dihydroindolone derivatives, method of preparing same and pharmaceutical compositions containing them SERVIER LAB (FR) 2013-01-16 EP disclosed
EP-2281822-A1 New dihydroindolone derivatives, method of preparing same and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2011-02-09 EP disclosed