SCHEMBL1228595

SCHEMBL1228595

CCC(C)(O)C#Cc1cc(Br)cnc1N

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 1/20 0.40
KMT2A Q03164 2/20 0.40
HTT P42858 1/20 0.40
TTBK1 Q5TCY1 7/20 0.38
TTBK2 Q6IQ55 4/20 0.38
MAP3K14 Q99558 3/20 0.38
HSD17B10 Q99714 3/20 0.34
KDM4E B2RXH2 2/20 0.34
NPC1 O15118 1/20 0.33
MEN1 O00255 1/20 0.31
PLA2G1B P04054 1/20 0.31
ATG4B Q9Y4P1 1/20 0.31
GAA P10253 1/20 0.31
DYRK1A Q13627 1/20 0.30
IDO1 P14902 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1204465 0.86 KMT2A (0.43) PGK1KMT2AHTTTTBK1MAP3K14
SCHEMBL21963753 0.79 HSD17B10 (0.43) KMT2AHTTHSD17B10KDM4ENPC1
SCHEMBL2040558 0.74 KMT2A (0.50) KMT2AHTTHSD17B10KDM4ENPC1
SCHEMBL2637090 0.71 KMT2A (0.47) KMT2AHTTNPC1MEN1DYRK1A
SCHEMBL17203284 0.71 KMT2A (0.43) KMT2AHTTHSD17B10KDM4ENPC1
SCHEMBL17203338 0.71 KMT2A (0.43) PGK1KMT2AHTTNPC1MEN1
SCHEMBL18430532 0.70 KMT2A (0.46) KMT2AHTTHSD17B10KDM4ENPC1
SCHEMBL1565246 0.70 HTT (0.39) KMT2AHTTHSD17B10KDM4ENPC1
SCHEMBL18741016 0.69 TDP1 (0.41) KMT2AHTTNPC1MEN1
SCHEMBL1203529 0.68 CSF1R (0.39) PGK1TTBK1MAP3K14IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462116-A2 PROCESS FOR THE MANUFACTURE OF PHARMACEUTICALLY ACTIVE COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-06-13 EP disclosed
WO-2011015522-A2 PROCESS FOR THE MANUFACTURE OF PHARMACEUTICALLY ACTIVE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-02-10 WO disclosed