SCHEMBL12290132

SCHEMBL12290132

O=C1c2cc(OC(F)(F)F)ccc2-n2c1nc1ccncc1c2=O

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 14/20 0.66
TDO2 P48775 9/20 0.50
IDO2 Q6ZQW0 7/20 0.50
APAF1 O14727 2/20 0.48
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
MITF O75030 1/20 0.48
HSP90AA1 P07900 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48
CHRM5 P08912 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593709 0.85 IDO1 (0.72) IDO1TDO2IDO2APAF1MEN1
SCHEMBL4593605 0.81 IDO1 (0.64) IDO1TDO2IDO2APAF1MEN1
SCHEMBL12290150 0.80 TDO2 (0.70) IDO1TDO2IDO2APAF1MEN1
SCHEMBL12290214 0.80 IDO1 (0.55) IDO1TDO2IDO2APAF1MEN1
SCHEMBL12325626 0.80 IDO1 (0.55) IDO1TDO2IDO2APAF1MEN1
SCHEMBL12289968 0.79 IDO1 (0.71) IDO1TDO2IDO2APAF1MEN1
SCHEMBL4593926 0.79 IDO1 (1.00) IDO1TDO2IDO2APAF1MEN1
SCHEMBL12290211 0.79 IDO1 (0.57) IDO1TDO2IDO2APAF1MEN1
SCHEMBL12325627 0.76 IDO1 (0.57) IDO1TDO2IDO2APAF1MEN1
SCHEMBL19456415 0.76 IDO1 (1.00) IDO1TDO2IDO2APAF1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012987-B2 Indolo[2,1-b] quinazole-6,12-dione antimalarial compounds and methods of treating malaria therewith THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 2011-09-06 US disclosed
US-8012987-B2 Indolo[2,1-b] quinazole-6,12-dione antimalarial compounds and methods of treating malaria therewith THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 2011-09-06 US disclosed