SCHEMBL12295292

SCHEMBL12295292

Cc1ccc(C(C)(c2ccc(C)cc2)C2CCCN2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
RAB9A P51151 1/20 0.44
TSHR P16473 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.35
CHRM2 P08172 3/20 0.34
CHRM4 P08173 2/20 0.34
CHRM5 P08912 2/20 0.34
CHRM1 P11229 2/20 0.34
CHRM3 P20309 2/20 0.34
MAPT P10636 1/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
MKNK1 Q9BUB5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10326595 1.00 CYP1A2 (0.44) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL10326467 1.00 CYP1A2 (0.44) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL10326278 0.87 HPGD (0.45) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL10326277 0.87 HPGD (0.45) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL8354404 0.86 CYP1A2 (0.44) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL10326564 0.84 CYP1A2 (0.45) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL10326582 0.84 CYP2D6 (0.62) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL10326879 0.84 CYP1A2 (0.45) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL10326896 0.84 CYP2D6 (0.62) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL10327263 0.84 CYP2D6 (0.62) CYP1A2CYP2D6CYP2C19KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438989-B1 USE OF ASYMMETRIC HYDROGENATION CATALYST TAKASAGO PERFUMERY CO LTD (JP) 2016-04-13 EP disclosed
EP-2543437-A2 HOMOGENEOUS ASYMMETRIC HYDROGENATION CATALYST Takasago International Corporation (JP) 2013-01-09 EP disclosed
WO-2011108672-A2 HOMOGENEOUS ASYMMETRIC HYDROGENATION CATALYST 高砂香料工業株式会社 (JP) 2011-09-09 WO disclosed
WO-2010140636-A1 ASYMMETRIC HYDROGENATION CATALYST 高砂香料工業株式会社 (JP) 2010-12-09 WO disclosed