SCHEMBL10326896

SCHEMBL10326896

CC(c1ccccc1)(c1ccccc1)[C@@H]1CCCN1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.62
CYP1A2 P05177 3/20 0.62
CYP2C19 P33261 2/20 0.62
KDM4E B2RXH2 1/20 0.62
NPC1 O15118 1/20 0.62
HPGD P15428 1/20 0.62
MAPK1 P28482 1/20 0.62
RAB9A P51151 1/20 0.62
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
LMNA P02545 2/20 0.37
HRH1 P35367 1/20 0.37
SCN1A P35498 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37
TACR1 P25103 4/20 0.36
TP53 P04637 2/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 2/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10326582 1.00 CYP2D6 (0.62) CYP2D6CYP1A2CYP2C19KDM4ENPC1
SCHEMBL10327263 1.00 CYP2D6 (0.62) CYP2D6CYP1A2CYP2C19KDM4ENPC1
SCHEMBL3236521 0.95 CYP2D6 (0.56) CYP2D6CYP1A2CYP2C19KDM4ENPC1
SCHEMBL10326938 0.90 CYP2C19 (0.49) CYP2D6CYP1A2CYP2C19KDM4ENPC1
SCHEMBL12295122 0.90 CYP2C19 (0.49) CYP2D6CYP1A2CYP2C19KDM4ENPC1
SCHEMBL10326936 0.90 CYP2C19 (0.49) CYP2D6CYP1A2CYP2C19KDM4ENPC1
SCHEMBL12295125 0.90 KDM4E (0.51) CYP2D6CYP1A2CYP2C19KDM4ENPC1
SCHEMBL10326804 0.90 KDM4E (0.51) CYP2D6CYP1A2CYP2C19KDM4ENPC1
SCHEMBL10326597 0.90 KDM4E (0.51) CYP2D6CYP1A2CYP2C19KDM4ENPC1
SCHEMBL12295126 0.86 CYP1A2 (0.51) CYP2D6CYP1A2CYP2C19KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170107213-A1 SUBSTITUTED NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES, PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME AND APPLICATIONS OFANTITUMOR THEREOF ZHEJIANG UNIVERSITY (CN) 2017-04-20 US disclosed
EP-2438989-B1 USE OF ASYMMETRIC HYDROGENATION CATALYST TAKASAGO PERFUMERY CO LTD (JP) 2016-04-13 EP disclosed
US-9040738-B2 Intermediate compounds of tamiflu, methods of preparation and uses thereof SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2015-05-26 US disclosed
US-20140221662-A1 INTERMEDIATE COMPOUNDS OF TAMIFLU, METHODS OF PREPARATION AND USES THEREOF SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2014-08-07 US disclosed
US-8217204-B2 Catalyst for asymmetric hydrogenation TAKASAGO INTERNATIONAL CORPORATION (JP) 2012-07-10 US disclosed
US-20100324338-A1 CATALYST FOR ASYMMETRIC HYDROGENATION TAKASAGO INTERNATIONAL CORPORATION (JP) 2010-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100324338-A1 CATALYST FOR ASYMMETRIC HYDROGENATION H1-0, H1-5, ADH5 CYP2D6 1125/4885CYP1A2 1183/4885CYP2C19 2363/4885
US-20170107213-A1 SUBSTITUTED NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES, PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME AND APPLICATIONS OFANTITUMOR THEREOF AKT1, RELA, AKT3 CYP2D6 1245/4885CYP1A2 2205/4885CYP2C19 2072/4885
US-20140221662-A1 INTERMEDIATE COMPOUNDS OF TAMIFLU, METHODS OF PREPARATION AND USES THEREOF NNMT, FLT3, TPMT CYP2D6 155/4885CYP1A2 112/4885CYP2C19 56/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.