SCHEMBL12296332

SCHEMBL12296332

CCc1nc2cc(Cl)ccn2c1C=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.38
CYP2C19 P33261 3/20 0.38
CYP3A4 P08684 1/20 0.37
PARP1 P09874 1/20 0.36
FGFR3 P22607 1/20 0.34
KDR P35968 1/20 0.34
HDAC1 Q13547 2/20 0.34
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MAT2A P31153 1/20 0.33
POLB P06746 1/20 0.33
GABRA1 P14867 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA5 P31644 2/20 0.33
PTGER4 P35408 1/20 0.32
NR1I3 Q14994 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14685289 0.78 CYP2C9 (0.39) CYP2C9CYP2C19CYP3A4PARP1ALDH1A1
SCHEMBL12294859 0.78 ALDH1A1 (0.42) CYP2C9CYP2C19CYP3A4PARP1ALDH1A1
SCHEMBL20377218 0.77 ALDH1A1 (0.55) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL15767382 0.77 CYP2C9 (0.38) CYP2C9CYP2C19CYP3A4PARP1FGFR3
SCHEMBL15330883 0.73 ALDH1A1 (0.52) PARP1ALDH1A1KDM4ENPC1RAB9A
SCHEMBL13838190 0.73 GAA (0.34) PARP1ALDH1A1KDM4ENPC1RAB9A
SCHEMBL17590056 0.72 CYP2C9 (0.46) CYP2C9CYP2C19CYP3A4PARP1FGFR3
SCHEMBL15333053 0.70 ALDH1A1 (0.48) PARP1ALDH1A1KDM4ENPC1RAB9A
SCHEMBL16447538 0.70 CYP2C9 (0.53) CYP2C9CYP2C19CYP3A4ALDH1A1KDM4E
SCHEMBL7081174 0.69 DPP4 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547678-B1 ANTI-INFECTIVE COMPOUNDS PASTEUR INSTITUT KOREA (KR) 2016-03-16 EP disclosed
WO-2011113606-A1 ANTI-INFECTIVE COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2011-09-22 WO disclosed