SCHEMBL12309142

SCHEMBL12309142

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nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 17/20 1.00
NFKB2 Q00653 17/20 1.00
RELA Q04206 17/20 1.00
CLPX O76031 1/20 0.85
VCP P55072 1/20 0.85
NPC1 O15118 1/20 0.68
POLB P06746 1/20 0.68
MAPT P10636 1/20 0.68
HTT P42858 1/20 0.68
RAB9A P51151 1/20 0.68
NPSR1 Q6W5P4 1/20 0.68
GLS O94925 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12309144 0.93 NFKB1 (0.89) NFKB1NFKB2RELACLPXVCP
SCHEMBL12309165 0.93 NFKB1 (1.00) NFKB1NFKB2RELACLPXVCP
SCHEMBL18944112 0.92 NFKB1 (0.85) NFKB1NFKB2RELACLPXVCP
SCHEMBL11950378 0.92 NFKB1 (0.85) NFKB1NFKB2RELACLPXVCP
SCHEMBL12309143 0.92 NFKB1 (1.00) NFKB1NFKB2RELACLPXVCP
SCHEMBL12309166 0.92 NFKB1 (1.00) NFKB1NFKB2RELACLPXVCP
SCHEMBL26519341 0.92 NFKB1 (1.00) NFKB1NFKB2RELACLPXVCP
SCHEMBL11950396 0.91 NFKB1 (0.84) NFKB1NFKB2RELACLPXVCP
SCHEMBL18943972 0.91 NFKB1 (0.84) NFKB1NFKB2RELACLPXVCP
SCHEMBL12309169 0.91 NFKB1 (0.83) NFKB1NFKB2RELACLPXVCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170066797-A1 WITHAFERIN A ANALOGS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2017-03-09 US disclosed
US-20170066797-A1 WITHAFERIN A ANALOGS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2017-03-09 US disclosed
US-20110230551-A1 WITHAFERIN A ANALOGS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH 2011-09-22 US disclosed
US-20110230551-A1 WITHAFERIN A ANALOGS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH 2011-09-22 US disclosed
WO-2010030395-A2 WITHAFERIN A ANALOGS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2010-03-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170066797-A1 WITHAFERIN A ANALOGS AND USES THEREOF CYP51A1, HASPIN, NFATC1 NFKB1 676/4885NFKB2 754/4885RELA 4064/4885
US-20110230551-A1 WITHAFERIN A ANALOGS AND USES THEREOF CYP51A1, HASPIN, NFATC1 NFKB1 676/4885NFKB2 754/4885RELA 4064/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.