SCHEMBL12320437

SCHEMBL12320437

CCOP(=O)(O)c1ccc(-c2nc3cc(C(=O)c4ccccc4)ccc3[nH]2)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.39
ALDH1A1 P00352 4/20 0.39
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
CHEK2 O96017 1/20 0.38
METAP1 P53582 1/20 0.38
MAPT P10636 4/20 0.37
LMNA P02545 3/20 0.37
CYP2C9 P11712 3/20 0.37
KDM4E B2RXH2 2/20 0.37
CYP1A2 P05177 2/20 0.37
HTT P42858 2/20 0.37
MAPK1 P28482 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2D6 P10635 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12618409 0.91 ESR1 (0.40) ESR1ALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL12320786 0.86 ESR1 (0.45) ESR1ALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL18890640 0.78 ALDH1A1 (0.50) ESR1ALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL1801134 0.76 ESR1 (0.47) ESR1ALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL1799546 0.76 MAPT (0.50) ESR1ALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL1801701 0.75 ESR1 (0.43) ESR1ALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL1797688 0.74 CHEK2 (0.52) ESR1ALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL1799498 0.72 TP53 (0.48) ESR1ALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL1801947 0.71 ALDH1A1 (0.41) ESR1ALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL34467256 0.71 CHEK2 (0.64) ESR1ALDH1A1HPGDSMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1911755-B1 BENZOIMIDAZOLE COMPOUND CAPABLE OF INHIBITING PROSTAGLANDIN D SYNTHETASE TAIHO PHARMACEUTICAL CO LTD (JP) 2011-09-14 EP disclosed
EP-1911755-A1 BENZOIMIDAZOLE COMPOUND CAPABLE OF INHIBITING PROSTAGLANDIN D SYNTHETASE TAIHO PHARMACEUTICAL CO., LTD. (JP) 2008-04-16 EP disclosed