SCHEMBL123276

SCHEMBL123276

C=CCOC(=O)OC1=C(C)N(c2cccc(C(F)(F)F)c2)C(=O)NC1c1ccc(C#N)cc1S(=O)(=O)C(C)C

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 0.58
CYP2C9 P11712 4/20 0.54
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL124739 0.93 ELANE (0.68) ELANECYP2C9CYP2C19
SCHEMBL122060 0.93 ELANE (0.68) ELANECYP2C9CYP2C19
SCHEMBL121526 0.92 ELANE (0.59) ELANECYP2C9CYP2C19
SCHEMBL122954 0.91 ELANE (0.66) ELANECYP2C9CYP2C19
SCHEMBL123937 0.91 ELANE (0.56) ELANECYP2C9CYP2C19
SCHEMBL1155172 0.90 ELANE (0.64) ELANECYP2C9CYP2C19
SCHEMBL121095 0.89 ELANE (0.64) ELANECYP2C9CYP2C19
SCHEMBL123311 0.87 ELANE (0.57) ELANECYP2C9
SCHEMBL121094 0.82 ELANE (0.72) ELANECYP2C9CYP2C19
SCHEMBL18086969 0.82 ELANE (0.75) ELANECYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234985-B1 4-(4-CYANO-2-THIOARYL)DIHYDROPYRIMIDINONES AND USE THEREOF Bayer Pharma AG (DE) 2012-03-07 EP disclosed
EP-2234985-A1 4-(4-CYANO-2-THIOARYL)DIHYDROPYRIMIDINONES AND USE THEREOF Bayer Schering Pharma Aktiengesellschaft (DE) 2010-10-06 EP disclosed
WO-2009080199-A1 4-(4-CYANO-2-THIOARYL)DIHYDROPYRIMIDINONES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed