SCHEMBL12345263

SCHEMBL12345263

Oc1ccc(C2C=C2)cc1O

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
QDPR P09417 3/20 0.47
ALOX5 P09917 2/20 0.47
PTPN1 P18031 1/20 0.47
AR P10275 1/20 0.44
APP P05067 2/20 0.43
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
TRPA1 O75762 1/20 0.40
YWHAG P61981 1/20 0.39
LCK P06239 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
SLC22A12 Q96S37 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17030563 0.78 PTPN1 (0.31) QDPRALOX5PTPN1AR
SCHEMBL10282755 0.72 QDPR (0.73) QDPRALOX5PTPN1APPMEN1
SCHEMBL108606 0.72 QDPR (0.73) QDPRALOX5PTPN1APPMEN1
SCHEMBL15095470 0.69 MEN1 (0.50) ARMEN1GAAKMT2ACA1
SCHEMBL2719092 0.69 MEN1 (0.50) ARMEN1GAAKMT2ACA1
SCHEMBL21816756 0.69 AR (0.72) QDPRALOX5PTPN1ARAPP
SCHEMBL15259264 0.69 QDPR (0.57) QDPRALOX5PTPN1ARAPP
SCHEMBL12251167 0.69 QDPR (0.44) QDPRALOX5PTPN1ARAPP
SCHEMBL107972 0.69 QDPR (0.57) QDPRALOX5PTPN1ARAPP
SCHEMBL107998 0.69 MEN1 (0.56) QDPRALOX5PTPN1MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2016065-B1 1-(BENZO[D][1,3]DIOXOL-5-YL)-N-(PHENYL)CYCLOPROPANE-CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS FOR THE TREATMENT OF CYSTIC FIBROSIS VERTEX PHARMA (US) 2012-09-19 EP disclosed