SCHEMBL12366128

SCHEMBL12366128

[C-]#[N+]CC(=O)NC1CCCc2ccccc21

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.69
TSHR P16473 2/20 0.63
HPGD P15428 2/20 0.63
MEN1 O00255 1/20 0.60
KMT2A Q03164 1/20 0.60
HTT P42858 4/20 0.59
POLB P06746 2/20 0.58
DHODH Q02127 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
TAOK1 Q7L7X3 1/20 0.57
TAOK3 Q9H2K8 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
EPHX1 P07099 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2213195 0.85 ALDH1A1 (0.74) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL53323 0.82 ALDH1A1 (1.00) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL20990440 0.82 ALDH1A1 (0.74) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL606143 0.82 ALDH1A1 (1.00) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL3729153 0.82 ALDH1A1 (0.74) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL14414533 0.82 ALDH1A1 (0.74) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL659023 0.82 ALDH1A1 (0.74) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL4003611 0.82 ALDH1A1 (0.74) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL4009579 0.82 ALDH1A1 (0.74) ALDH1A1TSHRHPGDMEN1KMT2A
SCHEMBL7932159 0.82 ALDH1A1 (0.74) ALDH1A1TSHRHPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed