SCHEMBL12368205

SCHEMBL12368205

COc1ccc(C)cc1NC(=O)c1cc(Br)ccc1O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNMA1 Q12791 3/20 0.61
ALDH1A1 P00352 2/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61
STAT3 P40763 1/20 0.60
KDM4E B2RXH2 5/20 0.59
RXFP1 Q9HBX9 1/20 0.59
POLB P06746 6/20 0.58
HSD17B10 Q99714 3/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
TSHR P16473 2/20 0.58
MAPT P10636 6/20 0.57
GFER P55789 1/20 0.57
LMNA P02545 2/20 0.57
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
NPSR1 Q6W5P4 2/20 0.56
MCL1 Q07820 1/20 0.56
NPC1 O15118 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14363385 0.91 KCNMA1 (0.68) KCNMA1ALDH1A1STAT3KDM4EPOLB
SCHEMBL331767 0.87 MAPT (0.59) ALDH1A1KDM4ERXFP1POLBHSD17B10
SCHEMBL12368204 0.84 MAPT (0.76) KCNMA1KDM4ERXFP1POLBHSD17B10
SCHEMBL7765905 0.84 MAPT (0.60) KCNMA1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL14363413 0.83 MEN1 (0.62) KCNMA1ALDH1A1KDM4EPOLBHSD17B10
SCHEMBL330396 0.83 TMPRSS4 (0.59) ALDH1A1CYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL12368201 0.82 HSD17B10 (0.65) KCNMA1ALDH1A1STAT3KDM4EPOLB
SCHEMBL14363387 0.82 KCNMA1 (0.75) KCNMA1ALDH1A1KDM4EPOLBHSD17B10
SCHEMBL330440 0.80 HTT (0.56) KCNMA1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL12368184 0.80 KMT2A (0.80) KCNMA1ALDH1A1KDM4EPOLBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989498-B2 Immunosuppressants; autoimmune disease; organs transplantation; antiinflammatory agents; viricides; antiproliferative agents; antitumor, anticancer agents VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-08-02 US disclosed
US-7989498-B2 Immunosuppressants; autoimmune disease; organs transplantation; antiinflammatory agents; viricides; antiproliferative agents; antitumor, anticancer agents VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-08-02 US disclosed
US-7915255-B2 Metabolism-modulating agents and uses therefor VERVA PHARMACEUTICALS PTY LTD (AU) 2011-03-29 US disclosed
US-7915255-B2 Metabolism-modulating agents and uses therefor VERVA PHARMACEUTICALS PTY LTD (AU) 2011-03-29 US disclosed