SCHEMBL12372142

SCHEMBL12372142

CC(=O)c1cc(C)cc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPMT P51580 2/20 0.44
CA5A P35218 1/20 0.44
KDR P35968 1/20 0.40
CYP2A6 P11509 1/20 0.39
HCAR1 Q9BXC0 2/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
KCNK3 O14649 1/20 0.38
KCNK9 Q9NPC2 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 4/20 0.37
RAB9A P51151 4/20 0.37
NPC1 O15118 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HTT P42858 1/20 0.37
NLRP1 Q9C000 1/20 0.37
CNR2 P34972 2/20 0.37
CNR1 P21554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL111207 0.85 TPMT (0.59) TPMTCA5AKDRHCAR1LMNA
Hydrochloric Acid SCHEMBL28868737 0.83 TPMT (0.56) TPMTCA5AKDRHCAR1LMNA
SCHEMBL2624954 0.83 TPMT (0.55) TPMTCA5ACYP2A6HCAR1LMNA
SCHEMBL95695 0.83 TPMT (0.62) TPMTCA5ACYP2A6HCAR1LMNA
SCHEMBL2172128 0.82 TPMT (0.44) TPMTKDRHCAR1CES2CES1
SCHEMBL668260 0.82 TPMT (0.44) TPMTKDRHCAR1CES2CES1
SCHEMBL29912669 0.82 TPMT (0.44) TPMTKDRHCAR1CES2CES1
SCHEMBL2172133 0.82 TPMT (0.70) TPMTKDRHCAR1SMN1; SMN2CNR2
SCHEMBL22383502 0.80 PARP1 (0.50) TPMTKDRHCAR1CES2CES1
SCHEMBL14110107 0.80 TPMT (0.43) TPMTCA5AKDRHCAR1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9174969-B2 Indoline scaffold SHP-2 inhibitors and cancer treatment method UNIVERSITY OF SOUTH FLORIDA (US) 2015-11-03 US disclosed
US-20150239889-A1 PYRAZOLOPYRIMIDINE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2015-08-27 US disclosed
US-20110190315-A1 INDOLINE SCAFFOLD SHP-2 INHIBITORS AND CANCER TREATMENT METHOD UNIVERSITY OF SOUTH FLORIDA (US) 2011-08-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150239889-A1 PYRAZOLOPYRIMIDINE COMPOUND HIF1AN, EGLN2, EGLN3 TPMT 1953/4885CA5A 186/4885KDR 164/4885
US-20110190315-A1 INDOLINE SCAFFOLD SHP-2 INHIBITORS AND CANCER TREATMENT METHOD PTPN7, PTPN3, PTPN5 TPMT 2881/4885CA5A 1800/4885KDR 740/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.