SCHEMBL12372656

SCHEMBL12372656

COc1ccc(Oc2ccc(C(=O)c3ccc(C(C)=O)cc3)cc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.73
HPGD P15428 2/20 0.73
RAB9A P51151 2/20 0.73
PARP10 Q53GL7 2/20 0.61
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
RXFP1 Q9HBX9 2/20 0.61
LMNA P02545 1/20 0.61
MAPK1 P28482 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
ALDH1A1 P00352 2/20 0.56
GAA P10253 1/20 0.56
CES2 O00748 1/20 0.55
CES1 P23141 1/20 0.55
TUBB4A P04350 1/20 0.54
TUBB P07437 1/20 0.54
TUBA3C P0DPH7 1/20 0.54
TUBA1B P68363 1/20 0.54
TUBA4A P68366 1/20 0.54
TUBB4B P68371 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14407940 1.00 MAPT (0.73) MAPTHPGDRAB9APARP10MEN1
SCHEMBL14198677 1.00 MAPT (0.73) MAPTHPGDRAB9APARP10MEN1
SCHEMBL12372650 1.00 MAPT (0.73) MAPTHPGDRAB9APARP10MEN1
SCHEMBL9963642 0.94 MAPT (0.68) MAPTHPGDRAB9APARP10MEN1
SCHEMBL13599772 0.94 MAPT (0.83) MAPTHPGDRAB9APARP10MEN1
SCHEMBL755167 0.94 MAPT (0.83) MAPTHPGDRAB9APARP10MEN1
SCHEMBL24538828 0.92 PARP10 (0.70) MAPTHPGDRAB9APARP10MEN1
SCHEMBL14407949 0.92 PARP10 (0.70) MAPTHPGDRAB9APARP10MEN1
SCHEMBL17469590 0.92 PARP10 (0.70) MAPTHPGDRAB9APARP10MEN1
SCHEMBL19008826 0.92 PARP10 (0.70) MAPTHPGDRAB9APARP10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110206880-A1 HIGH TEMPERATURE MELT PROCESSABLE SEMI-CRYSTALLINE POLY(ARYL ETHER KETONE) CONTAINING A (4-HYDROXYPHENYL)PHTHALAZIN-1(2H)-ONE COMONOMER UNIT WANG YI-FENG 2011-08-25 US disclosed