SCHEMBL12376218

SCHEMBL12376218

COc1ccc(C2(c3cccc(-c4cncnc4)c3)COC(N)=N2)cc1C(F)(F)F

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.71
CTSD P07339 9/20 0.54
BACE2 Q9Y5Z0 3/20 0.51
KCNH2 Q12809 5/20 0.48
REN P00797 1/20 0.44
CTSE P14091 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL2284111 0.95 BACE1 (0.64) BACE1CTSDBACE2KCNH2REN
SCHEMBL7865137 0.94 BACE1 (0.69) BACE1CTSDBACE2KCNH2REN
SCHEMBL12376216 0.92 BACE1 (0.71) BACE1CTSDBACE2KCNH2REN
SCHEMBL7863696 0.90 BACE1 (0.62) BACE1CTSDBACE2KCNH2
SCHEMBL7872670 0.90 BACE1 (0.57) BACE1CTSDBACE2KCNH2REN
SCHEMBL7865201 0.90 BACE1 (0.57) BACE1CTSDBACE2KCNH2
SCHEMBL7872518 0.88 BACE1 (0.70) BACE1CTSDBACE2KCNH2
SCHEMBL7874076 0.87 BACE1 (0.74) BACE1CTSDBACE2KCNH2REN
Formic Acid SCHEMBL2281054 0.87 BACE1 (0.65) BACE1CTSDBACE2KCNH2REN
Formic Acid SCHEMBL2283150 0.85 BACE1 (0.52) BACE1CTSDBACE2KCNH2REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-B1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-11-14 EP disclosed
US-7989449-B2 4,5-dihydro-oxazol-2-yl amine derivatives HOFFMAN-LA ROCHE INC. (US) 2011-08-02 US disclosed
US-7989449-B2 4,5-dihydro-oxazol-2-yl amine derivatives HOFFMAN-LA ROCHE INC. (US) 2011-08-02 US disclosed