SCHEMBL12377461

SCHEMBL12377461

Cc1ccc(OCc2nc(N)nc(N)c2-c2ccc(Cl)c(Cl)c2)cc1C

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.74
CYP3A4 P08684 2/20 0.74
TP53 P04637 1/20 0.74
CYP2D6 P10635 1/20 0.74
CYP2C9 P11712 1/20 0.74
CYP2C19 P33261 1/20 0.74
SMN1; SMN2 Q16637 1/20 0.74
HIF1A Q16665 1/20 0.74
DHFR P00374 6/20 0.48
REN P00797 1/20 0.44
NCOA1 Q15788 1/20 0.44
NCOA3 Q9Y6Q9 1/20 0.44
HEXA P06865 1/20 0.43
HEXB P07686 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8737810 0.86 CYP1A2 (1.00) CYP1A2CYP3A4TP53CYP2D6CYP2C9
SCHEMBL14813163 0.86 CYP1A2 (0.86) CYP1A2CYP3A4TP53CYP2D6CYP2C9
SCHEMBL9999991 0.86 CYP1A2 (0.82) CYP1A2CYP3A4TP53CYP2D6CYP2C9
SCHEMBL14813234 0.84 CYP1A2 (0.63) CYP1A2CYP3A4TP53CYP2D6CYP2C9
SCHEMBL7534201 0.84 CYP1A2 (0.62) CYP1A2CYP3A4TP53CYP2D6CYP2C9
SCHEMBL6049470 0.80 CYP1A2 (0.57) CYP1A2CYP3A4TP53CYP2D6CYP2C9
Etoprine SCHEMBL3919 0.76 DHFR (0.70) CYP1A2CYP3A4TP53CYP2D6CYP2C9
Metoprine SCHEMBL3681 0.72 NPC1 (0.54) CYP1A2CYP3A4TP53CYP2D6CYP2C9
Metoprine SCHEMBL29463675 0.72 NPC1 (0.54) CYP1A2CYP3A4TP53CYP2D6CYP2C9
Metoprine SCHEMBL4529657 0.70 NPC1 (0.53) CYP1A2CYP3A4TP53CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7994184-B2 Small molecules that replace or agonize p53 function BUCK INSTITUTE (US) 2011-08-09 US disclosed