SCHEMBL12409243

SCHEMBL12409243

Oc1ccc(-c2cnc3c(NCc4ccncc4)nccn23)cc1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TTK P33981 13/20 0.57
ADORA3 P0DMS8 6/20 0.53
FYN P06241 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12409244 0.91 TTK (0.68) TTKADORA3
SCHEMBL12409289 0.89 TTK (0.56) TTKADORA3FYN
SCHEMBL12409259 0.88 TTK (0.55) TTKADORA3FYN
SCHEMBL12409282 0.88 TTK (0.55) TTKADORA3
SCHEMBL12409227 0.88 TTK (0.51) TTKADORA3FYN
SCHEMBL12409283 0.88 TTK (0.55) TTKADORA3
SCHEMBL12409271 0.87 TTK (0.56) TTKADORA3FYN
SCHEMBL12409229 0.86 TTK (0.51) TTKADORA3FYN
SCHEMBL14668729 0.85 TTK (0.53) TTKADORA3
SCHEMBL12409305 0.85 TTK (0.55) TTKADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS CYP3A5, HAVCR2, CYP3A43 TTK 3239/4885ADORA3 4222/4885FYN 3511/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.