SCHEMBL12409259

SCHEMBL12409259

Oc1ccc(-c2cnc3c(NCc4ccc(Cl)cc4)nccn23)cc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TTK P33981 11/20 0.55
ADORA3 P0DMS8 6/20 0.54
FLT3 P36888 1/20 0.48
ADORA2A P29274 1/20 0.46
FYN P06241 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
NFKB1 P19838 1/20 0.43
RAB9A P51151 1/20 0.43
NFKB2 Q00653 1/20 0.43
KMT2A Q03164 1/20 0.43
RELA Q04206 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12409289 0.90 TTK (0.56) TTKADORA3FLT3FYN
SCHEMBL12409282 0.89 TTK (0.55) TTKADORA3KDM4EMEN1ALDH1A1
SCHEMBL12409244 0.88 TTK (0.68) TTKADORA3FLT3KDM4EALDH1A1
SCHEMBL12409243 0.88 TTK (0.57) TTKADORA3FYN
SCHEMBL14668729 0.88 TTK (0.53) TTKADORA3FLT3MAPT
SCHEMBL12409312 0.87 ADORA3 (0.56) TTKADORA3FLT3FYNMAPT
SCHEMBL12409268 0.86 TTK (0.52) TTKADORA3FLT3KDM4EALDH1A1
SCHEMBL12409283 0.86 TTK (0.55) TTKADORA3MAPT
SCHEMBL12409305 0.86 TTK (0.55) TTKADORA3
SCHEMBL12409255 0.86 TTK (0.52) TTKADORA3FYNMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193131-B1 IMIDAZO[1,2-A]PYRAZINE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS SUCH AS HEPATITIS BIOFOCUS DPI LTD (GB) 2013-01-30 EP disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS CYP3A5, HAVCR2, CYP3A43 TTK 3239/4885ADORA3 4222/4885FLT3 1683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.