SCHEMBL12409265

SCHEMBL12409265

COc1ccc(-c2cnc3c(NCCS(N)(=O)=O)nccn23)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 14/20 0.47
FYN P06241 2/20 0.43
FLT3 P36888 1/20 0.42
PAX8 Q06710 2/20 0.40
AURKA O14965 1/20 0.39
JAK2 O60674 1/20 0.39
MAP4K4 O95819 1/20 0.39
INSR P06213 1/20 0.39
LCK P06239 1/20 0.39
LYN P07948 1/20 0.39
RET P07949 1/20 0.39
ROS1 P08922 1/20 0.39
SRC P12931 1/20 0.39
FER P16591 1/20 0.39
KDR P35968 1/20 0.39
SYK P43405 1/20 0.39
BLK P51451 1/20 0.39
RPS6KA3 P51812 1/20 0.39
PRKCD Q05655 1/20 0.39
BTK Q06187 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12409232 0.85 FYN (0.62) TTKFYNSYK
SCHEMBL3470277 0.85 FYN (0.54) TTKFYNFLT3SYK
SCHEMBL12409240 0.83 FYN (0.53) TTKFYN
SCHEMBL12409321 0.83 FYN (0.48) TTKFYNFLT3
SCHEMBL12409254 0.82 TTK (0.49) TTKFYN
SCHEMBL12409292 0.81 FYN (0.60) TTKFYN
SCHEMBL12409252 0.80 ZAP70 (0.48) TTKFYNPAX8
SCHEMBL12409242 0.79 TTK (0.56) TTKFYNFLT3PAX8LCK
SCHEMBL12409235 0.79 PAX8 (0.48) TTKFYNPAX8RET
SCHEMBL12409284 0.78 QPCT (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS CYP3A5, HAVCR2, CYP3A43 TTK 3239/4885FYN 3511/4885FLT3 1683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.