SCHEMBL1242057

SCHEMBL1242057

NCC(=O)N(C(=O)c1ccccc1)C(c1ccccc1)C(O)(c1cccnc1)c1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 11/20 0.56
KCNH2 Q12809 6/20 0.50
LMNA P02545 2/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
EPHX2 P34913 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP3A5 P20815 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTT P42858 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1242288 0.80 KCNA5 (0.70) KCNA5KCNH2LMNACYP3A4CYP1A2
SCHEMBL1242188 0.75 KCNA5 (0.62) KCNA5KCNH2LMNACYP3A4CYP3A5
SCHEMBL1242189 0.75 KCNA5 (0.62) KCNA5KCNH2LMNACYP3A4CYP3A5
SCHEMBL1242980 0.75 KCNA5 (0.65) KCNA5KCNH2LMNACYP3A4CYP1A2
SCHEMBL1242838 0.73 KCNA5 (0.62) KCNA5KCNH2LMNACYP2C9CYP2C19
SCHEMBL1242316 0.73 KCNA5 (1.00) KCNA5KCNH2CYP3A4
SCHEMBL1242561 0.72 KCNA5 (1.00) KCNA5KCNH2CYP2C9CYP2C19CYP3A4
SCHEMBL1242823 0.72 KCNA5 (0.67) KCNA5KCNH2LMNACYP3A4CYP1A2
SCHEMBL1242947 0.72 KCNA5 (0.67) KCNA5KCNH2LMNACYP3A4CYP1A2
SCHEMBL1242273 0.71 KCNA5 (0.56) KCNA5KCNH2LMNAEPHX2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7879839-B2 For treatment and prevention of cardiac arrhythmias; (+-)-2-Morpholin-4-yl-2-phenyl-1,1-dipyridin-3-yl-ethanol; (+-)-2-[(2-methoxyethyl)(methyl)amino]-2-phenyl-1,1-dipyridin-3-ylethanol MERCK SHARP & DOHME CORP. (US) 2011-02-01 US disclosed