SCHEMBL12423364

SCHEMBL12423364

CCOC(=O)c1c(C(C)C)nc2c(c1I)C(O)CC(C)(C)C2

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CETP P11597 18/20 0.45
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10196397 1.00 CETP (0.45) CETPLMNAGAAHTTCYP1A2
SCHEMBL10196405 0.87 CETP (0.47) CETP
SCHEMBL12424361 0.87 CETP (0.47) CETP
SCHEMBL12423599 0.87 CETP (0.45) CETP
SCHEMBL10238046 0.87 CETP (0.45) CETP
SCHEMBL12424359 0.86 LMNA (0.44) CETPLMNAGAAHTTCYP1A2
SCHEMBL10196400 0.86 LMNA (0.44) CETPLMNAGAAHTTCYP1A2
SCHEMBL663922 0.85 CETP (0.48) CETP
SCHEMBL15182452 0.85 CETP (0.48) CETP
SCHEMBL15182458 0.85 CETP (0.48) CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536733-B1 TRICYCLIC PYRIDINE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PREPARATION BOEHRINGER INGELHEIM INT (DE) 2014-11-26 EP disclosed
WO-2013024149-A1 CRYSTALLINE FORMS OF OCTAHYDRO-3H-SPIRO [FURO [3, 4-C] QUINOLINE -1, 4 '-PYRAN] -9-OL BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-02-21 WO disclosed
WO-2011101424-A1 TRICYCLIC PYRIDINE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PREPARATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-25 WO disclosed