SCHEMBL12425239

SCHEMBL12425239

BN1CCC2(CC[C@@H](NC(C)=O)c3ccccc32)CC1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCHR2 Q969V1 9/20 0.47
DRD2 P14416 2/20 0.45
SLC6A4 P31645 2/20 0.45
KCNH2 Q12809 1/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.38
HSD11B1 P28845 2/20 0.37
HSD11B2 P80365 1/20 0.36
ALOX15 P16050 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13000675 0.83 MCHR2 (0.44) MCHR2DRD2SLC6A4KCNH2
SCHEMBL13207758 0.83 MCHR2 (0.44) MCHR2DRD2SLC6A4KCNH2
SCHEMBL13001193 0.83 MCHR2 (0.44) MCHR2DRD2SLC6A4KCNH2
SCHEMBL2758090 0.83 MCHR2 (0.52) MCHR2DRD2SLC6A4KCNH2ALDH1A1
SCHEMBL13000505 0.83 MCHR2 (0.44) MCHR2DRD2SLC6A4KCNH2
SCHEMBL13000018 0.83 SIGMAR1 (0.51) MCHR2DRD2SLC6A4KCNH2
SCHEMBL240547 0.82 MCHR2 (0.46) MCHR2DRD2SLC6A4KCNH2HSD11B1
SCHEMBL2758104 0.82 MCHR2 (0.52) MCHR2DRD2SLC6A4KCNH2ALDH1A1
SCHEMBL240548 0.82 MCHR2 (0.46) MCHR2DRD2SLC6A4KCNH2HSD11B1
SCHEMBL2758065 0.82 MCHR2 (0.50) MCHR2DRD2SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003660-B2 Modulators of muscarinic receptors VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-08-23 US disclosed