SCHEMBL12425614

SCHEMBL12425614

CC(C)(C)OC(=O)N1CCCC2CN(C(=O)c3ccc(N)nc3)CC21

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.50
MTOR P42345 2/20 0.50
SPR P35270 1/20 0.42
ALOX5AP P20292 2/20 0.42
FEN1 P39748 2/20 0.42
UCHL1 P09936 2/20 0.41
HDAC1 Q13547 2/20 0.40
NPC1 O15118 1/20 0.40
TRPC6 Q9Y210 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
HRH2 P25021 1/20 0.39
HRH1 P35367 1/20 0.39
KMT5A Q9NQR1 1/20 0.39
HPGDS O60760 1/20 0.39
USP30 Q70CQ3 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
GPR119 Q8TDV5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12426766 0.94 PIK3CA (0.46) PIK3CAMTORSPRALOX5APFEN1
SCHEMBL12425408 0.86 PIK3CA (0.41) PIK3CAMTORALOX5APFEN1TRPC6
SCHEMBL12425779 0.86 KMT5A (0.43) PIK3CAMTORTRPC6KMT5A
SCHEMBL12425620 0.84 CYP3A4 (0.41) PIK3CAMTORHRH2HRH1MEN1
SCHEMBL12426765 0.82 KMT5A (0.39) PIK3CAMTORKMT5A
SCHEMBL12425803 0.80 DPP4 (0.43) PIK3CAMTORKMT5A
SCHEMBL2301926 0.79 HDAC1 (0.48) PIK3CAMTORSPRALOX5APFEN1
SCHEMBL2300794 0.78 HDAC1 (0.52) SPRHDAC1MEN1KMT2AGPR119
SCHEMBL1990029 0.77 KMT2A (0.57) MEN1KMT2AGPR119
SCHEMBL12425594 0.77 HDAC1 (0.46) PIK3CAMTORSPRHDAC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101409-A1 PYRROLOPYRIMIDINE COMPOUNDS AS INHIBITORS OF CDK4/6 NOVARTIS AG (CH) 2011-08-25 WO disclosed