SCHEMBL1242667

SCHEMBL1242667

CCC(CC)n1cc(C(=O)N[C@H](Cc2cccnc2)C(=O)OC)c(=O)c2cc(F)c(NC3CCCCC3)cc21

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 2/20 0.47
PDE10A Q9Y233 1/20 0.42
NLRP3 Q96P20 1/20 0.41
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CNR1 P21554 3/20 0.37
CNR2 P34972 3/20 0.37
S1PR3 Q99500 3/20 0.36
BRD4 O60885 1/20 0.36
TACR3 P29371 1/20 0.35
PKM P14618 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DHODH Q02127 1/20 0.35
KRAS P01116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1242617 0.99 MEN1 (0.46) MEN1KMT2AGAAPDE10ANLRP3
SCHEMBL4107168 0.94 MEN1 (0.47) MEN1KMT2AGAAPDE10AALDH1A1
Hydrochloric Acid SCHEMBL4103837 0.93 MEN1 (0.47) MEN1KMT2AGAAPDE10AALDH1A1
SCHEMBL1242669 0.82 MEN1 (0.46) MEN1KMT2AGAAPDE10AALDH1A1
Hydrochloric Acid SCHEMBL1242620 0.82 MEN1 (0.46) MEN1KMT2AGAAPDE10AALDH1A1
SCHEMBL1242668 0.82 MEN1 (0.47) MEN1KMT2AGAAPDE10AALDH1A1
Hydrochloric Acid SCHEMBL1242618 0.81 MEN1 (0.46) MEN1KMT2AGAAPDE10AALDH1A1
SCHEMBL1242497 0.78 MEN1 (0.54) MEN1KMT2AGAAPDE10AALDH1A1
SCHEMBL27635118 0.78 MEN1 (0.54) MEN1KMT2AGAAPDE10AALDH1A1
SCHEMBL27635197 0.76 MEN1 (0.47) MEN1KMT2AGAAPDE10AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7879878-B2 such as {2-[({[7-(cyclohexylamino)-6-fluoro-4-oxo-1-[(3S)-tetrahydrofuran-3-yl]-1,4-dihydroquinolin-3-yl}carbonyl)amino]ethyl}phosphonic acid, used as platelet aggregation inhibitor and purinergic receptor (P2Y12) inhibitors; therapy for circulatory diseases involving thrombosis via platelet aggregation ASTELLAS PHARMA INC. (JP) 2011-02-01 US disclosed