SCHEMBL1242668

SCHEMBL1242668

CCC(CC)n1cc(C(=O)N[C@@H](C(=O)O)C(C)c2cccnc2)c(=O)c2cc(F)c(NC3CCCCC3)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
GAA P10253 2/20 0.47
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
LMNA P02545 1/20 0.37
ADRB3 P13945 2/20 0.37
GPR132 Q9UNW8 1/20 0.35
PDE10A Q9Y233 2/20 0.34
FOXO1 Q12778 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HPGD P15428 1/20 0.34
TOP2A P11388 1/20 0.34
TOP2B Q02880 1/20 0.34
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1242618 0.99 MEN1 (0.46) MEN1KMT2AGAAKDM4EALDH1A1
SCHEMBL4107168 0.85 MEN1 (0.47) MEN1KMT2AGAAKDM4EALDH1A1
Hydrochloric Acid SCHEMBL4103837 0.84 MEN1 (0.47) MEN1KMT2AGAAKDM4EALDH1A1
SCHEMBL1242667 0.82 MEN1 (0.47) MEN1KMT2AGAAKDM4EALDH1A1
Hydrochloric Acid SCHEMBL1242617 0.81 MEN1 (0.46) MEN1KMT2AGAAKDM4EALDH1A1
SCHEMBL1242669 0.80 MEN1 (0.46) MEN1KMT2AGAAKDM4EALDH1A1
Hydrochloric Acid SCHEMBL1242620 0.79 MEN1 (0.46) MEN1KMT2AGAAKDM4EALDH1A1
SCHEMBL27635118 0.78 MEN1 (0.54) MEN1KMT2AGAAKDM4EALDH1A1
SCHEMBL1242497 0.78 MEN1 (0.54) MEN1KMT2AGAAKDM4EALDH1A1
SCHEMBL1242593 0.76 GAA (0.57) MEN1KMT2AGAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7879878-B2 such as {2-[({[7-(cyclohexylamino)-6-fluoro-4-oxo-1-[(3S)-tetrahydrofuran-3-yl]-1,4-dihydroquinolin-3-yl}carbonyl)amino]ethyl}phosphonic acid, used as platelet aggregation inhibitor and purinergic receptor (P2Y12) inhibitors; therapy for circulatory diseases involving thrombosis via platelet aggregation ASTELLAS PHARMA INC. (JP) 2011-02-01 US disclosed