SCHEMBL12428152

SCHEMBL12428152

CCc1ccc2c(c1)N(CCN1CCCCCC1)CCn1c-2c(C2CCCCC2)c2ccc(C(=O)O)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.44
MMP12 P39900 1/20 0.44
SCN9A Q15858 4/20 0.41
CCR3 P51677 5/20 0.37
NR1I2 O75469 5/20 0.35
KCNH2 Q12809 5/20 0.34
HRH3 Q9Y5N1 3/20 0.34
HTR1A P08908 1/20 0.34
SLC6A4 P31645 1/20 0.34
HRH1 P35367 1/20 0.34
CYP3A4 P08684 2/20 0.33
SCN5A Q14524 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CHRM2 P08172 1/20 0.32
CYP2D6 P10635 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
CHRM3 P20309 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12428238 1.00 PRKCA (0.44) PRKCAMMP12SCN9ACCR3NR1I2
SCHEMBL12428061 1.00 PRKCA (0.44) PRKCAMMP12SCN9ACCR3NR1I2
SCHEMBL12428162 0.94 PRKCA (0.43) PRKCAMMP12SCN9ACCR3NR1I2
SCHEMBL804229 0.92 PRKCA (0.46) PRKCAMMP12SCN9ANR1I2KCNH2
SCHEMBL12428156 0.92 PRKCA (0.43) PRKCAMMP12SCN9ACCR3NR1I2
SCHEMBL12428189 0.92 PRKCA (0.42) PRKCAMMP12SCN9ACCR3NR1I2
SCHEMBL12427971 0.90 PRKCA (0.45) PRKCAMMP12SCN9ANR1I2KCNH2
SCHEMBL803833 0.90 PRKCA (0.45) PRKCAMMP12SCN9ANR1I2KCNH2
SCHEMBL12427895 0.90 PRKCA (0.45) PRKCAMMP12SCN9ANR1I2KCNH2
SCHEMBL804612 0.90 PRKCA (0.45) PRKCAMMP12SCN9ANR1I2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed