SCHEMBL12428173

SCHEMBL12428173

CCCc1ccc2c(c1)N(CCN1CCCC(COC)C1)CCn1c-2c(C2CCCCC2)c2ccc(C(=O)O)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.40
MMP12 P39900 1/20 0.40
SCN9A Q15858 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
CHRNB2 P17787 2/20 0.33
CHRNB4 P30926 2/20 0.33
CHRNA3 P32297 2/20 0.33
CHRNA4 P43681 2/20 0.33
KCNH2 Q12809 6/20 0.33
CYP3A4 P08684 3/20 0.33
SCN5A Q14524 2/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
DRD3 P35462 1/20 0.33
NR1I2 O75469 4/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10283272 0.94 PRKCA (0.41) PRKCAMMP12SCN9ACHRNB2CHRNB4
SCHEMBL803917 0.94 PRKCA (0.41) PRKCAMMP12SCN9AKCNH2CYP3A4
SCHEMBL10283551 0.90 PRKCA (0.42) PRKCAMMP12SCN9ACHRNB2CHRNB4
SCHEMBL12428544 0.90 PRKCA (0.42) PRKCAMMP12SCN9ACHRNB2CHRNB4
SCHEMBL12428047 0.90 PRKCA (0.42) PRKCAMMP12SCN9ACHRNB2CHRNB4
SCHEMBL12428213 0.90 PRKCA (0.42) PRKCAMMP12SCN9AKCNH2DRD2
SCHEMBL12428162 0.90 PRKCA (0.43) PRKCAMMP12SCN9AKCNH2NR1I2
SCHEMBL12428040 0.89 PRKCA (0.41) PRKCAMMP12SCN9ACHRNB2CHRNB4
SCHEMBL12429167 0.89 PRKCA (0.41) PRKCAMMP12SCN9AKCNH2CYP3A4
SCHEMBL12429164 0.89 PRKCA (0.41) PRKCAMMP12CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed