SCHEMBL12429034

SCHEMBL12429034

O=C(O)c1ccc2c(C3CCCCC3)c3n(c2c1)CCOc1c(-c2ccncc2)cccc1-3

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.47
MMP12 P39900 1/20 0.47
SCN9A Q15858 6/20 0.39
CYP3A4 P08684 2/20 0.38
CYP2C19 P33261 2/20 0.38
NR1I2 O75469 1/20 0.38
HPGD P15428 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
KMO O15229 1/20 0.35
STIM1 Q13586 1/20 0.34
ORAI1 Q96D31 1/20 0.34
RORC P51449 1/20 0.33
UCHL1 P09936 1/20 0.33
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
S1PR1 P21453 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL774479 0.99 PRKCA (0.47) PRKCAMMP12SCN9ACYP3A4CYP2C19
SCHEMBL773877 0.93 PRKCA (0.52) PRKCAMMP12SCN9ANR1I2POLB
SCHEMBL804237 0.91 PRKCA (0.46) PRKCAMMP12SCN9ANR1I2HPGD
Hydrochloric Acid SCHEMBL771873 0.91 PRKCA (0.46) PRKCAMMP12SCN9ANR1I2HPGD
SCHEMBL774666 0.87 PRKCA (0.48) PRKCAMMP12SCN9ANR1I2KMO
SCHEMBL774624 0.85 PRKCA (0.50) PRKCAMMP12SCN9ACYP3A4NR1I2
SCHEMBL771845 0.85 PRKCA (0.51) PRKCAMMP12SCN9ACYP3A4CYP2C19
SCHEMBL772514 0.84 PRKCA (0.49) PRKCAMMP12SCN9ANR1I2HPGD
SCHEMBL773242 0.84 PRKCA (0.55) PRKCAMMP12SCN9ACYP3A4CYP2C19
SCHEMBL773902 0.83 PRKCA (0.50) PRKCAMMP12SCN9ANR1I2KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed