SCHEMBL12432208

SCHEMBL12432208

CCC[C@@H](CC=O)Nc1ccccc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 10/20 0.39
HDAC1 Q13547 10/20 0.39
HDAC2 Q92769 8/20 0.39
HDAC8 Q9BY41 5/20 0.39
HDAC4 P56524 3/20 0.39
HDAC7 Q8WUI4 3/20 0.39
HDAC10 Q969S8 3/20 0.39
HDAC11 Q96DB2 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC9 Q9UKV0 3/20 0.39
HDAC5 Q9UQL6 3/20 0.39
TAS1R3 Q7RTX0 3/20 0.38
TAS1R1 Q7RTX1 3/20 0.38
NCOR2 Q9Y618 4/20 0.33
CA1 P00915 2/20 0.33
KCNH2 Q12809 1/20 0.33
CA2 P00918 1/20 0.33
AOC3 Q16853 1/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29922632 0.82 HDAC3 (0.40) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL21799890 0.82 HDAC3 (0.40) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL20685224 0.80 KCNH2 (0.42) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL11415357 0.75 IDO1 (0.49) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL29922607 0.74 TLR8 (0.41) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL21799545 0.74 TLR8 (0.41) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL2312159 0.73 ALDH1A1 (0.42) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL2312151 0.73 ALDH1A1 (0.42) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL21799625 0.68 IDO1 (0.42) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL22692976 0.67 CYP1A2 (0.39) HDAC3HDAC1HDAC2HDAC8HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152674-B1 BENZIMIDAZOLONE CHYMASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2011-08-03 EP disclosed