SCHEMBL12433302

SCHEMBL12433302

BCc1ccc2c(Br)cccc2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.55
GRM5 P41594 1/20 0.43
KCNH2 Q12809 1/20 0.43
C1R P00736 2/20 0.35
KMT2A Q03164 1/20 0.35
CYP1A2 P05177 1/20 0.34
TYMS P04818 2/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CYSLTR2 Q9NS75 1/20 0.32
CYSLTR1 Q9Y271 1/20 0.32
NOS1 P29475 1/20 0.32
AXL P30530 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
GUSB P08236 1/20 0.31
CDK9 P50750 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2706604 0.83 BACE1 (0.56) BACE1GRM5KCNH2C1RKMT2A
SCHEMBL29923487 0.81 BACE1 (0.55) BACE1GRM5KCNH2C1RKMT2A
SCHEMBL24695125 0.81 BACE1 (0.55) BACE1GRM5KCNH2C1RKMT2A
SCHEMBL31434331 0.75 BACE1 (0.51) BACE1GRM5KCNH2CYP1A2TYMS
SCHEMBL18995270 0.75 BACE1 (0.60) BACE1GRM5KCNH2C1RKMT2A
SCHEMBL28415013 0.74 BACE1 (0.64) BACE1GRM5KCNH2C1RKMT2A
SCHEMBL12152293 0.74 KCNH2 (0.57) BACE1KCNH2KDM4EALDH1A1GAA
SCHEMBL3067674 0.71 BACE1 (1.00) BACE1GRM5KCNH2TYMSKDM4E
SCHEMBL4953591 0.71 BACE1 (0.60) BACE1GRM5KCNH2C1RKMT2A
SCHEMBL707745 0.71 BACE1 (0.66) BACE1GRM5KCNH2C1RKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996180-B1 BENZAMIDE AND PYRIDYLAMIDE DERIVATIVES AS ANTIBACTERIAL AGENTS BIOTA EUROPE LTD (GB) 2011-08-03 EP disclosed