SCHEMBL29923487

SCHEMBL29923487

CCc1ccc2c(Br)cccc2n1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.55
GRM5 P41594 1/20 0.43
KCNH2 Q12809 1/20 0.43
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
ELANE P08246 3/20 0.36
KMT2A Q03164 2/20 0.35
C1R P00736 2/20 0.35
PARP1 P09874 1/20 0.35
CYP1A2 P05177 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
TYMS P04818 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24695125 1.00 BACE1 (0.55) BACE1GRM5KCNH2KDM4EALDH1A1
SCHEMBL2706604 0.83 BACE1 (0.56) BACE1GRM5KCNH2KDM4EALDH1A1
SCHEMBL12433302 0.81 BACE1 (0.55) BACE1GRM5KCNH2KDM4EALDH1A1
SCHEMBL12152293 0.80 KCNH2 (0.57) BACE1KCNH2KDM4EALDH1A1GAA
SCHEMBL4820896 0.78 HTR3A (0.46) BACE1KCNH2KDM4EALDH1A1GAA
SCHEMBL13668629 0.78 PDE10A (0.47) KDM4EALDH1A1GAAHPGDELANE
SCHEMBL6212842 0.78 KDM4E (0.47) BACE1KDM4EALDH1A1GAAHPGD
SCHEMBL17179176 0.78 PDE3B (0.41) KDM4EALDH1A1GAAHPGDELANE
SCHEMBL17179433 0.76 KDM4E (0.40) KDM4EALDH1A1GAAHPGDELANE
SCHEMBL18905189 0.75 ELANE (0.41) KDM4EALDH1A1GAAHPGDELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed