SCHEMBL12436925

SCHEMBL12436925

Cc1cc(-c2c[nH]c(C3[C@H]4CC[C@H](C4)N3C(=O)OC(C)(C)C)n2)ccc1-c1ncc(-c2c[nH]c([C@@H]3[C@H]4CC[C@H](C4)N3C(=O)OC(C)(C)C)n2)cc1C

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PREP P48147 2/20 0.36
JAK1 P23458 2/20 0.34
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
GPR119 Q8TDV5 3/20 0.32
RET P07949 2/20 0.32
JAK2 O60674 1/20 0.32
TYK2 P29597 1/20 0.32
JAK3 P52333 1/20 0.32
EIF2AK4 Q9P2K8 1/20 0.32
KCNK3 O14649 4/20 0.32
KCNK9 Q9NPC2 4/20 0.32
KAT2B Q92831 1/20 0.32
PIK3CA P42336 3/20 0.31
SUV39H2 Q9H5I1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12436928 0.86 PREP (0.41) PREPJAK1CHRM2CHRM1CHRM3
SCHEMBL12436556 0.86 PREP (0.41) PREPJAK1CHRM2CHRM1CHRM3
SCHEMBL16062569 0.85 PREP (0.40) PREPJAK1CHRM2CHRM1CHRM3
SCHEMBL12436385 0.84 PREP (0.42) PREPJAK1CHRM2CHRM1CHRM3
SCHEMBL17066303 0.84 PREP (0.42) PREPJAK1CHRM2CHRM1CHRM3
SCHEMBL12436927 0.84 PREP (0.41) PREPJAK1CHRM2CHRM1CHRM3
SCHEMBL12436783 0.81 CYP3A4 (0.38)
SCHEMBL16062559 0.81 KCNK3 (0.41) PREPJAK1CHRM2CHRM1CHRM3
SCHEMBL18426928 0.81 KCNK3 (0.41) PREPJAK1CHRM2CHRM1CHRM3
SCHEMBL889338 0.81 KCNK3 (0.41) PREPJAK1CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011091532-A1 HEPATITIS C INHIBITOR COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-04 WO disclosed