SCHEMBL12439

SCHEMBL12439

CC[C@H]1CCCN(CCN2CCOC(C)C2)C1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.43
BCHE P06276 1/20 0.38
DRD1 P21728 2/20 0.36
PDK1 Q15118 1/20 0.35
DRD3 P35462 5/20 0.35
PIK3CD O00329 1/20 0.34
PIK3R2 O00459 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
PIK3R5 Q8WYR1 1/20 0.34
PIK3R3 Q92569 1/20 0.34
CARM1 Q86X55 1/20 0.33
PRMT6 Q96LA8 1/20 0.33
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18082887 0.84 SIGMAR1 (0.46) BCHEDRD1DRD3CARM1PRMT6
SCHEMBL12446 0.82 KDM1A (0.46) KDM1ADRD1PDK1PIK3CDPIK3R2
SCHEMBL12781 0.82 KDM1A (0.46) KDM1ADRD1PDK1PIK3CDPIK3R2
SCHEMBL12449672 0.82 KDM1A (0.46) KDM1ADRD1PDK1PIK3CDPIK3R2
SCHEMBL12234177 0.81 KDM1A (0.50) KDM1ADRD1PDK1DRD3PIK3CD
SCHEMBL18082862 0.80 KDM1A (0.49) KDM1ADRD1PDK1DRD3PIK3CD
SCHEMBL17277354 0.79 CYP1A2 (0.42) BCHE
SCHEMBL25111811 0.78 KDM1A (0.40) KDM1ADRD1PDK1DRD3PIK3CD
Fluoride SCHEMBL30329860 0.78 DRD4 (0.49) BCHEDRD1DRD3DRD2DRD4
SCHEMBL26770451 0.76 KDM1A (0.38) KDM1ADRD1PDK1DRD3PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058149-A1 TRICYCLIC PYRAZOL AMINE DERIVATIVES MERCK SERONO S.A. (CH) 2011-05-19 WO disclosed