SCHEMBL12440359

SCHEMBL12440359

N[C@@H]1CCCN(CCOc2ccc(-c3ccc(-c4ccc(Cl)cc4)cn3)cc2)C1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 11/20 0.61
CHRM1 P11229 4/20 0.54
HTR2A P28223 4/20 0.54
CYP2D6 P10635 1/20 0.54
HRH3 Q9Y5N1 6/20 0.48
LTA4H P09960 2/20 0.48
PTGS2 P35354 1/20 0.48
HRH2 P25021 1/20 0.47
HRH1 P35367 1/20 0.47
SIGMAR1 Q99720 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12441547 0.94 MCHR1 (0.57) MCHR1CHRM1HTR2ACYP2D6HRH3
SCHEMBL12440251 0.86 MCHR1 (0.78) MCHR1CHRM1HTR2ACYP2D6HRH3
SCHEMBL14039753 0.86 MCHR1 (0.78) MCHR1CHRM1HTR2ACYP2D6HRH3
SCHEMBL12440372 0.86 MCHR1 (0.74) MCHR1CHRM1HTR2ACYP2D6HRH3
SCHEMBL12440472 0.85 MCHR1 (0.77) MCHR1CHRM1HTR2ACYP2D6HRH3
SCHEMBL4527666 0.85 MCHR1 (0.78) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4527655 0.85 MCHR1 (0.78) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL13933578 0.84 MCHR1 (0.57) MCHR1CHRM1HTR2ACYP2D6HRH3
SCHEMBL12441099 0.81 MCHR1 (0.72) MCHR1CHRM1HTR2ACYP2D6HRH3
SCHEMBL12440511 0.81 HRH3 (0.73) MCHR1CHRM1HTR2ACYP2D6HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2357173-A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-08-17 EP disclosed