SCHEMBL12440372

SCHEMBL12440372

Clc1ccc(-c2ccc(-c3ccc(OCCN4CCC4)cc3)nc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 10/20 0.74
CHRM1 P11229 2/20 0.66
HTR2A P28223 2/20 0.66
CYP2D6 P10635 1/20 0.66
LTA4H P09960 3/20 0.60
PTGS2 P35354 1/20 0.60
HRH3 Q9Y5N1 5/20 0.55
ACHE P22303 1/20 0.53
CXCR1 P25024 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440251 0.97 MCHR1 (0.78) MCHR1CHRM1HTR2ACYP2D6LTA4H
SCHEMBL14039753 0.97 MCHR1 (0.78) MCHR1CHRM1HTR2ACYP2D6LTA4H
SCHEMBL12440472 0.96 MCHR1 (0.77) MCHR1CHRM1HTR2ACYP2D6LTA4H
SCHEMBL13933577 0.90 MCHR1 (0.71) MCHR1CHRM1HTR2ACYP2D6LTA4H
SCHEMBL12440309 0.90 MCHR1 (0.76) MCHR1CHRM1HTR2ACYP2D6LTA4H
SCHEMBL12440423 0.88 MCHR1 (0.78) MCHR1CHRM1HTR2ACYP2D6LTA4H
SCHEMBL12441520 0.87 MCHR1 (0.61) MCHR1CHRM1HTR2ACYP2D6LTA4H
SCHEMBL12441099 0.87 MCHR1 (0.72) MCHR1CHRM1HTR2ACYP2D6HRH3
SCHEMBL12440511 0.86 HRH3 (0.73) MCHR1CHRM1HTR2ACYP2D6LTA4H
SCHEMBL12440359 0.86 MCHR1 (0.61) MCHR1CHRM1HTR2ACYP2D6LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2357173-A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-08-17 EP disclosed