SCHEMBL12440672

SCHEMBL12440672

Clc1ccc(-c2ccc(-c3ccc4oc(CN5CCCC5)nc4c3)nc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
SOS1 Q07889 1/20 0.46
POLB P06746 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP2C19 P33261 1/20 0.45
MCHR1 Q99705 4/20 0.42
HTR2C P28335 2/20 0.42
TMEM97 Q5BJF2 3/20 0.41
HDAC6 Q9UBN7 1/20 0.40
F10 P00742 1/20 0.39
CNR2 P34972 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12441354 0.85 NPC1 (0.51) NPC1RAB9ASOS1POLBHTT
SCHEMBL2322397 0.82 MCHR1 (0.56) NPC1RAB9ASOS1CYP2D6MCHR1
SCHEMBL12440592 0.76 ALDH1A1 (0.54) HTTMCHR1HTR2CCNR2
SCHEMBL12440591 0.76 MCHR1 (0.52) NPC1RAB9ACYP2D6CYP2C19MCHR1
SCHEMBL12440034 0.76 KDM4E (0.60) CYP2D6CYP2C19MCHR1HTR2CCNR2
SCHEMBL12440381 0.76 MCHR1 (0.52) NPC1RAB9APOLBHTTSMN1; SMN2
SCHEMBL2328403 0.72 NPC1 (0.46) NPC1RAB9ASOS1POLBHTT
SCHEMBL12440005 0.71 HRH3 (0.55) RAB9AMCHR1HRH3
SCHEMBL2328520 0.71 PIM1 (0.47) NPC1RAB9ASOS1SMN1; SMN2HDAC6
SCHEMBL4508812 0.71 SOS1 (0.45) NPC1RAB9ASOS1HTTTMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2357173-A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-08-17 EP disclosed