SCHEMBL12440740

SCHEMBL12440740

Fc1cc(Cl)ccc1-c1ccc(-c2ccc(OCCN3CCCC3)cc2)nn1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 5/20 0.61
LTA4H P09960 5/20 0.52
PTGS2 P35354 1/20 0.52
ACHE P22303 2/20 0.52
CYP2D6 P10635 1/20 0.47
CHRM1 P11229 1/20 0.47
HTR2A P28223 1/20 0.47
HRH3 Q9Y5N1 6/20 0.47
CXCR1 P25024 1/20 0.47
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440469 0.86 MCHR1 (0.78) MCHR1LTA4HPTGS2ACHECYP2D6
SCHEMBL13920751 0.86 MCHR1 (0.72) MCHR1LTA4HPTGS2ACHECYP2D6
SCHEMBL12440457 0.82 MCHR1 (0.59) MCHR1LTA4HPTGS2ACHECYP2D6
SCHEMBL30226262 0.77 MCHR1 (0.50) MCHR1LTA4HPTGS2HTR2A
SCHEMBL12440423 0.76 MCHR1 (0.78) MCHR1LTA4HPTGS2ACHECYP2D6
SCHEMBL2326926 0.76 MCHR1 (1.00) MCHR1LTA4HPTGS2CYP2D6CHRM1
SCHEMBL14039753 0.76 MCHR1 (0.78) MCHR1LTA4HPTGS2ACHECYP2D6
SCHEMBL12440251 0.76 MCHR1 (0.78) MCHR1LTA4HPTGS2ACHECYP2D6
SCHEMBL12440472 0.75 MCHR1 (0.77) MCHR1LTA4HPTGS2ACHECYP2D6
SCHEMBL7819691 0.74 LTA4H (0.90) LTA4HPTGS2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2357173-A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-08-17 EP disclosed