SCHEMBL12445579

SCHEMBL12445579

CC1(c2cc(NC(=O)c3ncccc3F)ccc2F)CC(=O)NC(N)=N1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.60
CYP2D6 P10635 1/20 0.48
BACE2 Q9Y5Z0 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12303291 0.83 BACE1 (0.60) BACE1CYP2D6BACE2
SCHEMBL12446176 0.81 BACE1 (0.57) BACE1BACE2
SCHEMBL12445623 0.81 BACE1 (0.53) BACE1BACE2
SCHEMBL1976782 0.80 BACE1 (0.73) BACE1CYP2D6BACE2
SCHEMBL4077508 0.80 BACE1 (0.72) BACE1BACE2
SCHEMBL4088227 0.79 BACE1 (0.77) BACE1BACE2
SCHEMBL1173322 0.79 BACE1 (0.81) BACE1BACE2
SCHEMBL2588183 0.79 BACE1 (0.71) BACE1CYP2D6BACE2
SCHEMBL12445836 0.77 BACE1 (0.49) BACE1BACE2
Formic Acid SCHEMBL2592659 0.76 BACE1 (0.67) BACE1CYP2D6BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2360155-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY Shionogi & Co., Ltd. (JP) 2011-08-24 EP disclosed