Formic Acid

Formic Acid

SCHEMBL2592659

C[C@@]1(c2cc(NC(=O)c3ncccc3F)ccc2F)CCOCC(N)=N1.O=CO

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.67
APP P05067 1/20 0.53
CYP2D6 P10635 1/20 0.53
BACE2 Q9Y5Z0 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2588183 0.96 BACE1 (0.71) BACE1APPCYP2D6BACE2
SCHEMBL1173322 0.88 BACE1 (0.81) BACE1APPBACE2
SCHEMBL2587828 0.85 BACE1 (0.78) BACE1APPBACE2
Formic Acid SCHEMBL2594420 0.85 BACE1 (0.67) BACE1BACE2
Formic Acid SCHEMBL15467301 0.85 BACE1 (0.67) BACE1BACE2
Formic Acid SCHEMBL2592575 0.84 BACE1 (0.93) BACE1APPBACE2
SCHEMBL1976782 0.84 BACE1 (0.73) BACE1CYP2D6BACE2
SCHEMBL15703753 0.82 BACE1 (0.64) BACE1APPBACE2
SCHEMBL2588794 0.82 BACE1 (0.84) BACE1APPCYP2D6BACE2
SCHEMBL2594490 0.81 BACE1 (0.71) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138293-A1 2,5,6,7-TETRAHYDRO-[1,4]OXAZEPIN-3-YLAMINE OR 2,3,6,7-TETRAHYDRO-[1,4]OXAZEPIN-5-YLAMINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-11-10 WO disclosed