SCHEMBL12445669

SCHEMBL12445669

Cc1noc(C)c1-c1cnc(C(=O)Nc2ccnc(C3(C)CC(=O)NC(N)=N3)c2)cn1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.40
AURKA O14965 3/20 0.39
AURKB Q96GD4 3/20 0.39
CYP2C8 P10632 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12301418 0.86 BACE1 (0.53) BACE1AURKAAURKB
SCHEMBL12445801 0.83 NPC1 (0.44) BACE1
SCHEMBL12445667 0.83 BACE1 (0.55) BACE1
SCHEMBL12445785 0.80 BACE1 (0.51) BACE1
SCHEMBL12445678 0.80 BACE1 (0.42) BACE1
SCHEMBL12445791 0.77 BACE1 (0.47) BACE1KCNH2
SCHEMBL12446242 0.76 BACE1 (0.44) BACE1
SCHEMBL12446250 0.74 BACE1 (0.48) BACE1AURKA
SCHEMBL7942055 0.74 BACE1 (0.71) BACE1
SCHEMBL12446238 0.74 BACE1 (0.56) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2360155-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY Shionogi & Co., Ltd. (JP) 2011-08-24 EP disclosed