SCHEMBL12445845

SCHEMBL12445845

Cc1c(C(=O)Nc2ccc(F)c(C3(C)CC(=O)NC(N)=N3)c2)oc2ccc(O)cc12

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.53
MAPT P10636 4/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
BACE2 Q9Y5Z0 1/20 0.41
HCRTR1 O43613 1/20 0.41
PPARG P37231 1/20 0.41
NCOR2 Q9Y618 1/20 0.41
APP P05067 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7933972 0.85 BACE1 (0.52) BACE1MAPTKDM4EALDH1A1GAA
SCHEMBL12446176 0.79 BACE1 (0.57) BACE1BACE2
SCHEMBL7943380 0.78 BACE1 (0.53) BACE1MAPTKDM4EALDH1A1GAA
SCHEMBL12302218 0.78 BACE1 (0.53) BACE1MAPTKDM4EALDH1A1GAA
SCHEMBL7942669 0.77 BACE1 (0.54) BACE1BACE2
SCHEMBL7943378 0.77 BACE1 (0.62) BACE1MAPTKDM4EALDH1A1GAA
SCHEMBL7944886 0.76 BACE1 (0.52) BACE1BACE2
SCHEMBL7944999 0.75 BACE1 (0.54) BACE1MAPTKDM4EALDH1A1BACE2
SCHEMBL12445623 0.75 BACE1 (0.53) BACE1BACE2
SCHEMBL12445579 0.74 BACE1 (0.60) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2360155-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY Shionogi & Co., Ltd. (JP) 2011-08-24 EP disclosed