SCHEMBL12463000

SCHEMBL12463000

Bc1cn2nc(C=O)nc2c(N2CCOCC2)n1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 1/20 0.36
POLB P06746 2/20 0.36
PIK3CA P42336 4/20 0.33
PIK3R1 P27986 3/20 0.33
MTOR P42345 3/20 0.33
PIK3CD O00329 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
KDM4E B2RXH2 3/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPT P10636 2/20 0.32
PDE10A Q9Y233 1/20 0.32
ALDH3A1 P30838 1/20 0.31
ALDH1A3 P47895 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14725941 0.84 ALDH1A1 (0.37) ALDH1A1L3MBTL1GAAPOLBPIK3CA
SCHEMBL12462791 0.79 ALDH1A1 (0.39) ALDH1A1GAAPOLBPIK3CAPIK3R1
SCHEMBL12462793 0.75 PDE4A (0.36) ALDH1A1GAAPOLBPIK3CAPIK3R1
SCHEMBL14725985 0.68 KDM4E (0.43) ALDH1A1L3MBTL1POLBKDM4EMEN1
SCHEMBL13896917 0.65 PIK3CA (0.45) PIK3CAPIK3R1MTORPIK3CDPIK3CB
SCHEMBL12463396 0.64 POLB (0.39) ALDH1A1GAAPOLBPIK3CAPIK3R1
SCHEMBL14149150 0.63 KDM4E (0.63) ALDH1A1GAAPOLBKDM4EMEN1
SCHEMBL5561919 0.62 HTR2C (0.39) ALDH1A1L3MBTL1GAAPOLBPIK3CA
SCHEMBL14725935 0.62 ALDH1A1 (0.39) ALDH1A1POLBPIK3CAPIK3R1KDM4E
SCHEMBL26071904 0.61 KDM4E (0.39) ALDH1A1L3MBTL1POLBPIK3CAPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011089400-A1 INHIBITORS OF PI3 KINASE CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2011-07-28 WO disclosed