SCHEMBL12464440

SCHEMBL12464440

CC1CC(C(=O)N(c2cc(-c3ccccc3)sc2C(=O)O)C2CCN(C)CC2)C1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.40
OPRM1 P35372 2/20 0.37
NR1I2 O75469 2/20 0.37
KDM4E B2RXH2 2/20 0.36
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.36
CACNA2D1 P54289 1/20 0.36
SCN1A P35498 1/20 0.35
SCN2A Q99250 1/20 0.35
SCN3A Q9NY46 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2873417 0.92 NR1I2 (0.44) MKNK1OPRM1NR1I2KDM4EHTT
SCHEMBL102095 0.92 NR1I2 (0.44) MKNK1OPRM1NR1I2KDM4EHTT
Hydrochloric Acid SCHEMBL2876957 0.91 NR1I2 (0.43) MKNK1OPRM1NR1I2KDM4EHTT
Hydrochloric Acid SCHEMBL2876954 0.91 NR1I2 (0.43) MKNK1OPRM1NR1I2KDM4EHTT
SCHEMBL12464670 0.89 KDM4E (0.38) OPRM1KDM4EHTTATM
SCHEMBL2876653 0.89 NR1I2 (0.46) MKNK1OPRM1NR1I2KDM4EHTT
Hydrochloric Acid SCHEMBL2871152 0.88 NR1I2 (0.45) MKNK1OPRM1NR1I2KDM4EHTT
SCHEMBL12464253 0.87 KDM4E (0.37) KDM4EHTTATM
SCHEMBL2876758 0.85 NR1I2 (0.42) MKNK1OPRM1NR1I2CACNA2D1
SCHEMBL2874205 0.84 NR1I2 (0.43) OPRM1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7985769-B2 Compounds and methods for the treatment or prevention of Flavivirus infections VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-07-26 US disclosed