SCHEMBL12465259

SCHEMBL12465259

Cc1ccc(NC(=O)c2cc(N3CCN(C)CC3)cc(C(F)(F)F)c2)cc1-n1cc(-c2cncs2)nn1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRAF P15056 12/20 0.59
CSF1R P07333 2/20 0.57
RAF1 P04049 2/20 0.57
LYN P07948 1/20 0.57
TEK Q02763 2/20 0.56
HCK P08631 1/20 0.49
NR2C2 P49116 1/20 0.49
BTK Q06187 1/20 0.49
ABL1 P00519 2/20 0.48
BCR P11274 2/20 0.48
GPR142 Q7Z601 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12398541 0.91 BRAF (0.59) BRAFCSF1RLYNHCKNR2C2
SCHEMBL12465255 0.87 BRAF (0.67) BRAFCSF1RRAF1LYNTEK
SCHEMBL12465254 0.87 ABL1 (0.52) BRAFABL1BCR
SCHEMBL12465258 0.87 ABL1 (0.52) BRAFABL1BCR
SCHEMBL12465141 0.86 BRAF (0.57) BRAFCSF1RRAF1LYNTEK
SCHEMBL13960025 0.85 CSF1R (0.56) BRAFCSF1RRAF1LYNTEK
SCHEMBL12465028 0.85 BRAF (0.64) BRAFCSF1RRAF1LYNTEK
SCHEMBL12465257 0.85 BRAF (0.57) BRAFCSF1RRAF1LYNTEK
SCHEMBL12464983 0.83 ABL1 (0.50) BRAFCSF1RTEKABL1BCR
SCHEMBL12398499 0.83 ABL1 (0.55) BRAFABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889665-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-18 US disclosed
US-20110183952-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110183952-A1 NEW CHEMICAL COMPOUNDS MKI67, CCNA1, CCNT1 BRAF 525/4885CSF1R 594/4885RAF1 394/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.