SCHEMBL12467244

SCHEMBL12467244

NC(=O)OCc1ccc(N2CCC(c3cc(C(F)(F)F)cc(C(F)(F)F)c3)(C(F)(F)F)C2O)nc1Br

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.32
USP2 O75604 2/20 0.31
CYP3A4 P08684 2/20 0.31
TSHR P16473 1/20 0.31
HIF1A Q16665 1/20 0.31
CYP2D6 P10635 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
AOC3 Q16853 1/20 0.30
ADAM17 P78536 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL794066 0.86
SCHEMBL807885 0.86
SCHEMBL12467308 0.83 TRPV1 (0.36) TACR1
SCHEMBL794134 0.82 TRPV1 (0.37) TACR1
SCHEMBL795181 0.81 CACNA1H (0.39) TACR1TSHRCYP2D6
SCHEMBL12467053 0.80 CYP3A4 (0.33) TACR1USP2CYP3A4TSHRHIF1A
SCHEMBL794562 0.67 AR (0.31)
SCHEMBL794922 0.65 KCNH2 (0.37)
SCHEMBL15474193 0.64 TRPV1 (0.36)
SCHEMBL795090 0.64 TRPV1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616437-A1 PESTICIDAL ARYLPYRROLIDINES Bayer Intellectual Property GmbH (DE) 2013-07-24 EP disclosed
WO-2012035011-A1 PESTICIDAL ARYLPYRROLIDINES BAYER CROPSCIENCE AG (DE) 2012-03-22 WO disclosed