SCHEMBL12469870

SCHEMBL12469870

CCOc1ccc2c(c1)OC(C)(C)CC21C(=O)N(Cc2ccc(F)cc2C#N)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 11/20 0.41
CYP3A4 P08684 1/20 0.35
MAOB P27338 3/20 0.35
ALDH1A1 P00352 2/20 0.33
CTSD P07339 1/20 0.33
BACE1 P56817 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CHRM1 P11229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469992 0.91 SCN9A (0.43) SCN9ACYP3A4MAOBALDH1A1CTSD
SCHEMBL12470200 0.87 SCN9A (0.41) SCN9ACYP3A4MAOBALDH1A1
SCHEMBL12469858 0.85 SCN9A (0.45) SCN9ACYP3A4MAOBMAPT
SCHEMBL12470330 0.84 MAOB (0.47) SCN9ACYP3A4MAOBMAPT
SCHEMBL12470231 0.83 MAOB (0.46) SCN9ACYP3A4MAOBALDH1A1CTSD
SCHEMBL12470006 0.82 SCN9A (0.42) SCN9ACYP3A4MAOBALDH1A1
SCHEMBL12470315 0.82 MAPT (0.42) SCN9ACYP3A4MAOBALDH1A1CTSD
SCHEMBL12470256 0.80 SCN9A (0.51) SCN9ACYP3A4MAPT
SCHEMBL12470007 0.79 SCN9A (0.50) SCN9ACYP3A4MAOBCTSDBACE1
SCHEMBL12470044 0.79 SCN9A (0.44) SCN9ACYP3A4MAOBALDH1A1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012049555-A1 SPIROCYCLIC COMPOUNDS AS VOLTAGE-GATED SODIUM CHANNEL MODULATORS LUPIN LIMITED (IN) 2012-04-19 WO claimed